EAU 2026: Phase 1/2 Study of an Anti-PD-L1/IL-15 Variant Fusion Protein (SIM0237) in BCG Unresponsive High-Risk NMIBC

(UroToday.com) The 2026 European Association of Urology (EAU) annual meeting featured a high-risk non-muscle invasive bladder cancer session and a presentation by Dr. Dingwei Ye discussing results of a phase 1/2 study of an anti-PD-L1/IL-15 variant fusion protein (SIM0237) in BCG unresponsive high-risk non-muscle invasive bladder cancer.

Treatment options for BCG-unresponsive non-muscle invasive bladder cancer are limited. Anti-PD-1 monotherapy and IL-15 agonist in combination with BCG have shown clinical efficacy in BCG-unresponsive CIS non-muscle invasive bladder cancer. However, it remains unclear whether targeting both PD-(L)1 and IL-15 has a synergistic effect in non-muscle invasive bladder cancer. SIM0237 is an anti-PD-L1/IL-15 variant fusion protein, which has shown a good safety profile and promising efficacy signal in patients with BCG-unresponsive non-muscle invasive bladder cancer in the dose escalation part of this trial:

 

At EAU 2026, Dr. Ye and colleagues reported data from the dose escalation and expansion parts of SIM0237 monotherapy from this ongoing phase 1/2 study.

Patients with BCG-unresponsive high-risk non-muscle invasive bladder cancer received intravesical SIM0237 following the standard induction + maintenance treatment schedule. A re-induction course was allowed if the patients had persistent CIS or high-grade Ta at month 3. Key study endpoints included dose-limiting toxicity, safety, tolerability, pharmacokinetics, and efficacy, defined as (i) the complete response rate and duration of complete response for CIS non-muscle invasive bladder cancer, or (ii) disease-free survival and disease-free survival rate at specific time points for papillary-only non muscle invasive bladder cancer:

Patients with BCG-unresponsive high-risk non-muscle invasive bladder cancer received intravesical SIM0237 following the standard induction + maintenance treatment schedule. A re-induction course was allowed if the patients had persistent CIS or high-grade Ta at month 3. Key study endpoints included dose limiting toxicity, safety, tolerability, pharmacokinetics and efficacy, defined as (i) the complete response rate and duration of complete response for CIS non muscle invasive bladder cancer, or (ii) disease free survival and disease free survival rate at specific time points for papillary-only non muscle invasive bladder cancer: 

From January 10, 2024, to the data cutoff date of November 28, 2025, a total of 49 patients (14 CIS with or without Ta/T1, 35 papillary-only) have received SIM0237 monotherapy. In the CIS with or without papillary group, the median age was 63 years (range: 51-73), with 78.6% male, and a median number of prior BCG doses of 13.5 (range: 5-30). In the papillary only group, the median age was 63 years (range: 36-87), with 77.1% male, and a median number of prior BCG doses of 13 (range: 6-46):

 From January 10, 2024, to the data cutoff date of November 28, 2025, a total of 49 patients (14 CIS with or without Ta/T1, 35 papillary-only) have received SIM0237 monotherapy. In the CIS with or without papillary group, the median age was 63 years (range: 51-73), with 78.6% male, and a median number of prior BCG doses of 13.5 (range: 5-30). In the papillary only group, the median age was 63 years (range: 36-87), with 77.1% male, and a median number of prior BCG doses of 13 (range: 6-46): 

The median follow-up was 6.7 months (range: 0-20.8 months). Of the 10 CIS patients who had at least 1 post-baseline tumor assessment, 8 achieved a best response of complete response, with a median duration of complete response immature, and a probability of duration of complete response 12+ months of 71.4% (95% CI 25.8-92.0%): 

The median follow-up was 6.7 months (range: 0-20.8 months). Of the 10 CIS patients who had at least 1 post-baseline tumor assessment, 8 achieved a best response of complete response, with a median duration of complete response immature, and a probability of duration of complete response 12+ months of 71.4% (95% CI 25.8-92.0%):  

In the 35 papillary-only patients, the median disease-free survival was immature, with a 12-month disease-free survival rate of 65.8% (95% CI, 44.1%-80.7%):

In the 35 papillary-only patients, the median disease-free survival was immature, with a 12-month disease-free survival rate of 65.8% (95% CI, 44.1%-80.7%): 

Treatment-emergent adverse events occurred in 42 (85.7%) patients, and 25 (51.0%) patients had treatment-related adverse events. The majority of treatment-related adverse events were grade 1/2 and limited to the urinary system. Overall, there were 10 (20.4%) patients who had grade 3+ treatment-emergent adverse events and 1 (2.0%) grade 3+ treatment-related adverse event. No grade 4 or 5 treatment emergent adverse events were reported. Four (8.2%) patients had serious adverse events, and 1 (2.0%) had a treatment-related serious adverse event of urinary bladder hemorrhage and prostatic hemorrhage. Eleven (22.4%) patients had dose interruptions due to treatment-emergent adverse events, and 5 (10.2%) had dose interruptions due to treatment-related adverse events. There were no dose-limiting toxicities, immune-related adverse events, or adverse events leading to SIM0237 discontinuation. Pharmacokinetics data showed undetectable systemic exposure of SIM0237 in all 29 patients with serum samples analyzed: 

Treatment-emergent adverse events occurred in 42 (85.7%) patients, and 25 (51.0%) patients had treatment-related adverse events. The majority of treatment-related adverse events were grade 1/2 and limited to the urinary system. Overall, there were 10 (20.4%) patients who had grade 3+ treatment-emergent adverse events and 1 (2.0%) grade 3+ treatment-related adverse event. No grade 4 or 5 treatment emergent adverse events were reported. Four (8.2%) patients had serious adverse events, and 1 (2.0%) had a treatment-related serious adverse event of urinary bladder hemorrhage and prostatic hemorrhage. Eleven (22.4%) patients had dose interruptions due to treatment-emergent adverse events, and 5 (10.2%) had dose interruptions due to treatment-related adverse events. There were no dose-limiting toxicities, immune-related adverse events, or adverse events leading to SIM0237 discontinuation. Pharmacokinetics data showed undetectable systemic exposure of SIM0237 in all 29 patients with serum samples analyzed:  

Dr. Ye concluded this presentation discussing results of a phase 1/2 study of SIM0237 in BCG-unresponsive high-risk non-muscle invasive bladder cancer with the following take-home points:

  • Intravesical SIM0237 was safe and well-tolerated, with promising clinical efficacy in patients with BCG-unresponsive high-risk non-muscle invasive bladder cancer
  • A phase 3 study of SIM0237 monotherapy in this patient population is being planned 

Presented by: Dingwei Ye, Professor, Fudan University Shanghai Cancer Center, Shanghai, China

Written by: Zachary Klaassen, MD, MSc – Urologic Oncologist, Associate Professor of Urology, Georgia Cancer Center, Wellstar MCG Health, @zklaassen_md on Twitter during the 2026 European Association of Urology (EAU) Annual Meeting, London, United Kingdom, Fri, Mar 13 – Mon, Mar 16, 2026.